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Amino Acid

Glycine

The smallest amino acid and an inhibitory neurotransmitter that improves sleep quality by lowering core body temperature through peripheral vasodilation. Beyond sleep, glycine is a rate-limiting substrate for glutathione synthesis and — paired with N-acetylcysteine — has reversed multiple hallmarks of aging in human trials (the GlyNAC research).

sleeplongevitycognitive-healthmetabolic-health
Tier AWell-tolerated — strong human evidence
Evidence gradeBControlled trials / Cohort studies
BH

Reviewed & fact-checked by

BiohackingHub Research Team

Editorial Research Team · Last updated: May 8, 2026

Verified

Stacking Interactions

How Glycine interacts with other compounds

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ApigeninSynergisticmoderate evidence

Glycine lowers core temperature for sleep onset while apigenin acts on GABA-A — two distinct sleep-onset mechanisms that combine well.

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L-TheanineSynergisticmoderate evidence

L-theanine reduces sleep-onset anxiety and glutamatergic excitation; glycine handles thermoregulatory sleep onset — non-overlapping and complementary.

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Magnesium ThreonateSynergisticmoderate evidence

Magnesium supports GABAergic tone and NMDA regulation; with glycine it rounds out a deep-sleep architecture stack.

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NMNSynergisticweak evidence

Glycine supports glutathione and methylation balance; pairs with NAD+ precursors in longevity-oriented stacks.

Safety Profile — Tier A

Well-tolerated — strong human evidence

Contraindications

  • Clozapine therapy — glycine may reduce clozapine efficacy
  • Rare inborn errors of glycine metabolism

Side Effects

  • Very well-tolerated; doses of 3-90g/day used in trials
  • Mild GI upset or loose stool at high single doses (uncommon)
  • Slight drowsiness when taken before bed (intended effect)

Drug Interactions

Clozapine — glycine antagonizes its therapeutic NMDA effectNo other clinically significant interactions reported